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Cisatracurium Besylate Injection 5ml:10mg
Composition:
Each 5ml vial contains:
- Cisatracurium Besylate ......… 10mg
Description:
Cisatracurium Besylate is a non-depolarizing neuromuscular blocking agent used as an adjunct to general anesthesia to facilitate endotracheal intubation and provide skeletal muscle relaxation during surgery or mechanical ventilation. It has intermediate duration and is metabolized by Hofmann elimination, making it suitable for patients with hepatic or renal impairment.
Indications:
- Facilitation of endotracheal intubation
- Skeletal muscle relaxation during surgery
- Mechanical ventilation in intensive care settings
Dosage & Administration:
For IV Use Only.
- Initial Dose for Intubation: 0.15-0.2 mg/kg IV bolus
- Maintenance Dose: 0.03 mg/kg IV as needed
- Continuous Infusion: 1-3 mcg/kg/min IV
Administration:
- Administer only by trained healthcare professionals
- Monitor neuromuscular function closely
- Use a peripheral nerve stimulator to guide dosing
Contraindications:
- Hypersensitivity to Cisatracurium or other neuromuscular blocking agents
Warnings & Precautions:
- Must be administered in a controlled setting with ventilatory support available
- Can cause respiratory paralysis - ensure ventilatory assistance
- Caution in patients with neuromuscular disorders (e.g., myasthenia gravis)
- Histamine release is minimal, but hypersensitivity reactions can occur
Adverse Reactions:
- Common: Hypotension, flushing, mild bradycardia
- Serious: Prolonged neuromuscular blockade, anaphylaxis
Drug Interactions:
- Enhanced effect with inhaled anesthetics (e.g., isoflurane, sevoflurane)
- Potentiated by aminoglycosides, magnesium, lithium
- Reduced effect by anticonvulsants (phenytoin, carbamazepine)
Storage Conditions:
- Store at 2°C-8°C (36°F-46°F) (Refrigerated)
- Protect from light
- Do not freeze


