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Linezolid and Glucose Injection 100ml:0.2g
Composition:
Each 100ml contains:
- Linezolid 0.2g (200mg)
- Glucose (sufficient quantity)
Description:
Linezolid is an oxazolidinone-class antibiotic with activity against Gram-positive bacteria, including resistant strains like methicillin-resistant Staphylococcus aureus (MRSA) and vancomycin-resistant enterococci (VRE). The glucose component provides necessary caloric intake for patients requiring parenteral nutrition support.
Indications:
Linezolid and Glucose Injection is indicated for the treatment of infections caused by susceptible Gram-positive bacteria, including:
- Nosocomial pneumonia (including MRSA-related pneumonia)
- Community-acquired pneumonia
- Complicated skin and soft tissue infections
- Vancomycin-resistant Enterococcus faecium (VRE) infections, including bacteremia
Dosage & Administration:
Adults & Adolescents (≥12 years):
- 600mg IV every 12 hours (infused over 30-120 minutes)
- Duration: 10-14 days, depending on infection severity
Pediatric Patients (<12 years):
- 10 mg/kg IV every 8 hours
- Duration: 10-14 days
Administration:
- Intravenous (IV) infusion only
- Administer over 30-120 minutes
- Do NOT mix with other IV medications
- No further dilution required
Contraindications:
- Hypersensitivity to Linezolid or any component of the formulation
- Patients using monoamine oxidase inhibitors (MAOIs) or within 2 weeks of MAOI use
Precautions:
- Myelosuppression (thrombocytopenia, anemia, leukopenia) - Monitor CBC weekly.
- Peripheral & optic neuropathy - Prolonged use may cause vision problems.
- Serotonin Syndrome Risk - Avoid with SSRIs, SNRIs, or other serotonergic drugs.
- Lactic Acidosis - Monitor for unexplained acidosis or low bicarbonate levels.
- Hyperglycemia risk - Caution in diabetic patients due to glucose content.
Adverse Reactions:
- Hematologic: Thrombocytopenia, anemia
- Neurologic: Headache, peripheral neuropathy
- Gastrointestinal: Nausea, vomiting, diarrhea
- Metabolic: Lactic acidosis, hyperglycemia
- Injection Site Reactions: Phlebitis, irritation
Drug Interactions:
- SSRIs, SNRIs, Tricyclic Antidepressants - Increased serotonin syndrome risk
- MAOIs (e.g., phenelzine, isocarboxazid) - Risk of hypertensive crisis
- Adrenergic agents (e.g., pseudoephedrine) - May enhance hypertensive effects
- Hypoglycemic agents (e.g., insulin) - Monitor blood glucose levels
Storage Conditions:
- Store below 25°C, protect from light.
- Do NOT freeze.
- Use within 24 hours after opening.
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